Download App
Home › Glossary

Peptide, GLP-1 & pharmacokinetics glossary

Plain-English definitions of the terms behind every compound profile and calculator on Halflife Labs — from half-life and steady state to reconstitution and titration. Each term links to the relevant tool or compound data.

Half-life (t½)
The time it takes for the active concentration of a compound in the bloodstream to fall by 50%. It governs dosing frequency and how long a compound stays in your system. Model any compound's decay with the half-life calculator or browse values in the compound database.
Steady state
The equilibrium reached when the amount of a compound entering the body equals the amount being cleared, so concentrations plateau. It typically takes about 4–5 half-lives of consistent dosing. See how to calculate steady state.
Cmax (peak concentration)
The maximum plasma concentration a compound reaches after a dose. Higher Cmax can mean stronger peak effects and, for some compounds, more pronounced side effects shortly after injection.
Tmax (time to peak)
The time after administration at which Cmax (peak concentration) occurs. Tmax depends on the route of administration and the compound's absorption rate.
Trough
The lowest concentration of a compound in the dosing interval, reached just before the next dose. The days-5–7 trough on weekly GLP-1s is why some users feel effects fade before their next injection.
AUC (area under the curve)
A measure of total compound exposure over time, calculated as the area under the concentration-versus-time curve. AUC reflects how much active compound the body is exposed to across the whole interval.
Elimination / clearance
The processes by which the body removes a compound, mainly via the kidneys (renal), liver (hepatic), and enzymatic breakdown. Clearance rate, together with dose, determines steady-state concentration.
First-order kinetics
Elimination in which a constant fraction (not a fixed amount) of the compound is cleared per unit time. Most peptides and GLP-1 medications follow first-order kinetics, which is what makes half-life a meaningful, constant value.
Bioavailability
The fraction of an administered dose that reaches systemic circulation in active form. Intravenous dosing is 100% by definition; subcutaneous, intramuscular, oral, and intranasal routes are typically lower.
Protein (albumin) binding
The reversible attachment of a compound to plasma proteins such as albumin. High albumin binding (as engineered into tirzepatide and several long-acting insulins) dramatically extends half-life by shielding the compound from clearance.
Reconstitution
Dissolving a lyophilised (freeze-dried) peptide with a diluent — usually bacteriostatic water — to create an injectable solution at a known concentration. Get exact volumes with the reconstitution calculator.
Bacteriostatic water (BAC)
Sterile water containing 0.9% benzyl alcohol, which inhibits bacterial growth and allows a reconstituted vial to be used over multiple days. It is the standard diluent for reconstituting peptides.
Subcutaneous (SC) injection
An injection into the fatty layer just under the skin, the most common route for peptides and GLP-1 medications. Rotating sites prevents tissue damage — track it with the injection site rotation tracker.
Titration / dose escalation
Gradually increasing a dose over weeks to improve tolerability, standard for GLP-1 medications. Build a personalised schedule with the GLP-1 dose escalation calculator.
Ester
A chemical group attached to a hormone (such as testosterone) to slow its release and extend half-life. Longer esters like cypionate and enanthate allow less frequent injections. See testosterone cypionate.
GLP-1 receptor agonist
A class of compounds that activate the GLP-1 receptor to reduce appetite and improve glycaemic control, including semaglutide and tirzepatide (a dual GIP/GLP-1 agonist).
GH secretagogue
A compound that stimulates the body's own release of growth hormone, rather than supplying GH directly. Includes GHRH analogues like CJC-1295 and ghrelin-mimetics like ipamorelin.
Lipohypertrophy
Lumps of thickened tissue caused by repeatedly injecting the same site, which impairs absorption. Rotating injection sites prevents it — see the rotation tracker.

Put these terms into practice

Halflife turns half-life, steady state, and trough into a live concentration curve for your own protocol. Free on iOS.

Download on the App Store
Or browse all 44 compounds →